Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein Dimerization

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Main Authors: Ioannis Gkekas, Katerina Pliatsika, Stelios Mylonas, Sotirios Katsamakas, Apostolos Axenopoulos, Simona Kostova, Erich E. Wanker, Dimitra Hadjipavlou-Litina, Konstantinos Xanthopoulos, Petros Daras, Spyros Petrakis
Format: Article
Language:English
Published: American Chemical Society 2025-06-01
Series:ACS Omega
Online Access:https://doi.org/10.1021/acsomega.5c02465
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author Ioannis Gkekas
Katerina Pliatsika
Stelios Mylonas
Sotirios Katsamakas
Apostolos Axenopoulos
Simona Kostova
Erich E. Wanker
Dimitra Hadjipavlou-Litina
Konstantinos Xanthopoulos
Petros Daras
Spyros Petrakis
author_facet Ioannis Gkekas
Katerina Pliatsika
Stelios Mylonas
Sotirios Katsamakas
Apostolos Axenopoulos
Simona Kostova
Erich E. Wanker
Dimitra Hadjipavlou-Litina
Konstantinos Xanthopoulos
Petros Daras
Spyros Petrakis
author_sort Ioannis Gkekas
collection DOAJ
format Article
id doaj-art-c4ca45a89dfa4e048df1cfd42d6f26d1
institution Kabale University
issn 2470-1343
language English
publishDate 2025-06-01
publisher American Chemical Society
record_format Article
series ACS Omega
spelling doaj-art-c4ca45a89dfa4e048df1cfd42d6f26d12025-08-20T03:29:07ZengAmerican Chemical SocietyACS Omega2470-13432025-06-011025271942720510.1021/acsomega.5c02465Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein DimerizationIoannis Gkekas0Katerina Pliatsika1Stelios Mylonas2Sotirios Katsamakas3Apostolos Axenopoulos4Simona Kostova5Erich E. Wanker6Dimitra Hadjipavlou-Litina7Konstantinos Xanthopoulos8Petros Daras9Spyros Petrakis10Institute of Applied Biosciences, Centre for Research and Technology Hellas, Thessaloniki, GreeceInstitute of Applied Biosciences, Centre for Research and Technology Hellas, Thessaloniki, GreeceInformation Technologies Institute, Centre for Research and Technology Hellas, Thessaloniki, GreeceLaboratory of Pharmaceutical Chemistry, School of Pharmacy, Faculty of Health Sciences, Aristotle University of Thessaloniki, Thessaloniki, GreeceInformation Technologies Institute, Centre for Research and Technology Hellas, Thessaloniki, GreeceMax-Delbrueck-Center for Molecular Medicine in the Helmholtz Association, Berlin, GermanyMax-Delbrueck-Center for Molecular Medicine in the Helmholtz Association, Berlin, GermanyLaboratory of Pharmaceutical Chemistry, School of Pharmacy, Faculty of Health Sciences, Aristotle University of Thessaloniki, Thessaloniki, GreeceInstitute of Applied Biosciences, Centre for Research and Technology Hellas, Thessaloniki, GreeceInformation Technologies Institute, Centre for Research and Technology Hellas, Thessaloniki, GreeceInstitute of Applied Biosciences, Centre for Research and Technology Hellas, Thessaloniki, Greecehttps://doi.org/10.1021/acsomega.5c02465
spellingShingle Ioannis Gkekas
Katerina Pliatsika
Stelios Mylonas
Sotirios Katsamakas
Apostolos Axenopoulos
Simona Kostova
Erich E. Wanker
Dimitra Hadjipavlou-Litina
Konstantinos Xanthopoulos
Petros Daras
Spyros Petrakis
Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein Dimerization
ACS Omega
title Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein Dimerization
title_full Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein Dimerization
title_fullStr Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein Dimerization
title_full_unstemmed Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein Dimerization
title_short Chemical Targeting of the ATXN1 aa99–163 Interaction Site Suppresses polyQ-Expanded Protein Dimerization
title_sort chemical targeting of the atxn1 aa99 163 interaction site suppresses polyq expanded protein dimerization
url https://doi.org/10.1021/acsomega.5c02465
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