A Robust Regression-Based Modeling to Predict Antiplasmodial Activity of Thiazolyl–Pyrimidine Hybrid Derivatives against <i>Plasmodium falciparum</i>
Thiazolyl–pyrimidine hybrid plays significant roles in the biological activities and SAR of thiazolylpyrimidines (Tzpd), thiazolopyrimidines, and thienopyrimidines due to the combination of the thiazole and pyrimidine pharmacophores. The study developed regression-based models for the prediction of...
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| Main Authors: | Kevin S. Umoette, Charles O. Nnadi, Wilfred O. Obonga |
|---|---|
| Format: | Article |
| Language: | English |
| Published: |
MDPI AG
2023-11-01
|
| Series: | Chemistry Proceedings |
| Subjects: | |
| Online Access: | https://www.mdpi.com/2673-4583/14/1/52 |
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