Rethinking MYC inhibition: a multi-dimensional approach to overcome cancer’s master regulator

MYC, a master regulator in oncogenesis, has long been deemed “undruggable” due to its intrinsically disordered structure. However, recent advances are overturning this view, with direct inhibitors like Omomyc (OMO-103) and PROTAC-based degraders such as WBC100 showing promising clinical progress. Co...

Full description

Saved in:
Bibliographic Details
Main Authors: Jing Yu, Dan Liu, Yujian Yuan, Chunxia Sun, Zihan Su
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-04-01
Series:Frontiers in Cell and Developmental Biology
Subjects:
Online Access:https://www.frontiersin.org/articles/10.3389/fcell.2025.1601975/full
Tags: Add Tag
No Tags, Be the first to tag this record!