Design, synthesis, and pharmacological evaluation of haloperidol derivatives as novel potent calcium channel blockers with vasodilator activity.

Several haloperidol derivatives with a piperidine scaffold that was decorated at the nitrogen atom with different alkyl, benzyl, or substituted benzyl moieties were synthesized at our laboratory to establish a library of compounds with vasodilator activity. Compounds were screened for vasodilatory a...

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Bibliographic Details
Main Authors: Yicun Chen, Jinhong Zheng, Fuchun Zheng, Jinzhi Wang, Yanmei Zhang, Fenfei Gao, Zhanqin Huang, Ganggang Shi
Format: Article
Language:English
Published: Public Library of Science (PLoS) 2011-01-01
Series:PLoS ONE
Online Access:https://journals.plos.org/plosone/article/file?id=10.1371/journal.pone.0027673&type=printable
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