Kinetics of endothelin-1 and effect selective ETA antagonism on ETB activation: a mathematical modeling analysis

IntroductionEndothelin-1 (ET-1) regulates renal and vascular function, but the clinical utility of selective ETA receptor antagonists has been limited due to associated fluid retention. The mechanisms underlying fluid retention remain poorly understood but could be a consequence of changes in ET-1 b...

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Bibliographic Details
Main Authors: K. Melissa Hallow, Peter J. Greasley, Hiddo J. L. Heerspink, Hongtao Yu
Format: Article
Language:English
Published: Frontiers Media S.A. 2024-11-01
Series:Frontiers in Pharmacology
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Online Access:https://www.frontiersin.org/articles/10.3389/fphar.2024.1332388/full
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