From In Vivo Predictive Dissolution to Virtual Bioequivalence: A GastroPlus<sup>®</sup>-Driven Framework for Generic Candesartan Cilexetil Tablets

<b>Background</b>: Candesartan cilexetil, a Biopharmaceutics Classification System (BCS) II prodrug, demonstrates compromised bioavailability attributable to its limited aqueous solubility coupled with P-glycoprotein (P-gp)-mediated efflux and hepatic first-pass metabolism, thereby intro...

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Bibliographic Details
Main Authors: Hao Ruan, Xiaoting Geng, Zijing Situ, Qian Shen, Tianjian Ye, Xin Chen, Weike Su
Format: Article
Language:English
Published: MDPI AG 2025-04-01
Series:Pharmaceuticals
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Online Access:https://www.mdpi.com/1424-8247/18/4/562
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