Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666

Two new decalin-tetramic acid hybrid metabolites, zopfiellamides C (<b>1</b>) and D (<b>2</b>) were isolated from the marine-derived fungus <i>Aspergillus</i> sp. NF666. The structure determination was accomplished on the basis of HRESIMS and NMR spectral data ana...

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Main Authors: Fangwen Jiao, Tianyu Liu, Kaiwei Wang, Shuai Li, Ruihua Jiao, Wei Lin
Format: Article
Language:English
Published: MDPI AG 2025-03-01
Series:Molecules
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Online Access:https://www.mdpi.com/1420-3049/30/7/1502
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author Fangwen Jiao
Tianyu Liu
Kaiwei Wang
Shuai Li
Ruihua Jiao
Wei Lin
author_facet Fangwen Jiao
Tianyu Liu
Kaiwei Wang
Shuai Li
Ruihua Jiao
Wei Lin
author_sort Fangwen Jiao
collection DOAJ
description Two new decalin-tetramic acid hybrid metabolites, zopfiellamides C (<b>1</b>) and D (<b>2</b>) were isolated from the marine-derived fungus <i>Aspergillus</i> sp. NF666. The structure determination was accomplished on the basis of HRESIMS and NMR spectral data analyses including COSY, HSQC, HMBC, and NOESY experiments. Both isolated metabolites (<b>1</b> and <b>2</b>) exhibited significant growth inhibition against four clinically relevant bacterial strains with minimum inhibitory concentration (MIC) values of about 12.5 μΜ. Moreover, we proposed a plausible biosynthetic pathway of zopfiellamide D (<b>2</b>) in this work.
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institution OA Journals
issn 1420-3049
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publishDate 2025-03-01
publisher MDPI AG
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series Molecules
spelling doaj-art-db8770f5f79b4aa89c0e94a874f127142025-08-20T02:17:01ZengMDPI AGMolecules1420-30492025-03-01307150210.3390/molecules30071502Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666Fangwen Jiao0Tianyu Liu1Kaiwei Wang2Shuai Li3Ruihua Jiao4Wei Lin5Department of Pathogen Biology, School of Medicine, Nanjing University of Chinese Medicine, Nanjing 210023, ChinaDepartment of Pathogen Biology, School of Medicine, Nanjing University of Chinese Medicine, Nanjing 210023, ChinaDepartment of Pathogen Biology, School of Medicine, Nanjing University of Chinese Medicine, Nanjing 210023, ChinaDepartment of Pathogen Biology, School of Medicine, Nanjing University of Chinese Medicine, Nanjing 210023, ChinaState Key Laboratory of Pharmaceutical Biotechnology, Institute of Functional Biomolecules, School of Life Sciences, Nanjing University, Nanjing 210023, ChinaDepartment of Pathogen Biology, School of Medicine, Nanjing University of Chinese Medicine, Nanjing 210023, ChinaTwo new decalin-tetramic acid hybrid metabolites, zopfiellamides C (<b>1</b>) and D (<b>2</b>) were isolated from the marine-derived fungus <i>Aspergillus</i> sp. NF666. The structure determination was accomplished on the basis of HRESIMS and NMR spectral data analyses including COSY, HSQC, HMBC, and NOESY experiments. Both isolated metabolites (<b>1</b> and <b>2</b>) exhibited significant growth inhibition against four clinically relevant bacterial strains with minimum inhibitory concentration (MIC) values of about 12.5 μΜ. Moreover, we proposed a plausible biosynthetic pathway of zopfiellamide D (<b>2</b>) in this work.https://www.mdpi.com/1420-3049/30/7/1502tetramic acidzopfiellamidesmarine fungus<i>Aspergillus</i> sp.structure elucidationantibacterial activity
spellingShingle Fangwen Jiao
Tianyu Liu
Kaiwei Wang
Shuai Li
Ruihua Jiao
Wei Lin
Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666
Molecules
tetramic acid
zopfiellamides
marine fungus
<i>Aspergillus</i> sp.
structure elucidation
antibacterial activity
title Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666
title_full Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666
title_fullStr Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666
title_full_unstemmed Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666
title_short Zopfiellamides C and D, New Decalin-Type Tetramic Acid Derivatives from the Marine-Derived Fungus <i>Aspergillus</i> sp. NF666
title_sort zopfiellamides c and d new decalin type tetramic acid derivatives from the marine derived fungus i aspergillus i sp nf666
topic tetramic acid
zopfiellamides
marine fungus
<i>Aspergillus</i> sp.
structure elucidation
antibacterial activity
url https://www.mdpi.com/1420-3049/30/7/1502
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