Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center Trial

Xue-Qi Li,1 Yang Liu,1 Ze-Yu Cai,1 Tie-Gang Lv,2 Jian Hao1 1Department of Medicine, Division of Nephrology, The Affiliated Hospital of Inner Mongolia Medical University, Hohhot, Inner Mongolia Autonomous Region, 010050, China; 2Department of Medicine, Division of Radiology, The Affiliated Hospital o...

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Main Authors: Li XQ, Liu Y, Cai ZY, Lv TG, Hao J
Format: Article
Language:English
Published: Dove Medical Press 2025-07-01
Series:Drug Design, Development and Therapy
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Online Access:https://www.dovepress.com/obinutuzumab-is-effective-as-an-initial-treatment-for-pla2r-associated-peer-reviewed-fulltext-article-DDDT
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author Li XQ
Liu Y
Cai ZY
Lv TG
Hao J
author_facet Li XQ
Liu Y
Cai ZY
Lv TG
Hao J
author_sort Li XQ
collection DOAJ
description Xue-Qi Li,1 Yang Liu,1 Ze-Yu Cai,1 Tie-Gang Lv,2 Jian Hao1 1Department of Medicine, Division of Nephrology, The Affiliated Hospital of Inner Mongolia Medical University, Hohhot, Inner Mongolia Autonomous Region, 010050, China; 2Department of Medicine, Division of Radiology, The Affiliated Hospital of Inner Mongolia Medical University, Hohhot, Inner Mongolia Autonomous Region, 010050, People’s Republic of ChinaCorrespondence: Jian Hao, Department of Medicine, Division of Nephrology, The Affiliated Hospital of Inner Mongolia Medical University, No. 1 North Passage Road, Huimin District, Hohhot, Inner Mongolia Autonomous Region, 010050, People’s Republic of China, Tel +8613704751021, Email jian_hao8865@126.comBackground: Membranous nephropathy (MN) can cause nephrotic syndrome. B cells contribute to MN, but available treatments are often inadequate. We addressed this treatment gap by analyzing the effect of obinutuzumab in patients with primary MN (PMN).Methods: Forty-seven PMN patients were followed for six months, with 25 receiving obinutuzumab and 22 (control) receiving rituximab. Treatment response was assessed by 24-h urine total protein (24-h UTP), serum albumin (ALB), and other indicators. Immunologic remission was assessed by measurement of anti-phospholipase A2 receptor autoantibodies (PLA2R autoAbs).Results: Relative to baseline, the obinutuzumab group had significant decreases of PLA2R autoAbs (83.40 [55.90– 344.36] vs 0.41 [0.17– 1.20] RU/mL), 24-h UTP (8.90 [7.15– 13.80) vs 1.82 [1.12– 3.43] g/day), and B cells (312.61 [202.00– 406.12) vs 0 [0– 0] cells/μL), and a significant increase of serum ALB (25.90 [20.85– 28.70] vs 42 [39.7– 45.3] g/L) after six months. Nineteen of the evaluable patients (76% [55– 91%]) achieved immunological remission at three months, 20 (80% [60– 93%] achieved immunological remission at six months, and 16 (64% [42– 83%] achieved partial response (PR) at three-months. After six-months, no patients achieved complete remission, but 19 (76% [55– 91%]) achieved PR. Before the second dose of obinutuzumab, the CD19+ B cell count in 20 patients (80%) [60%– 93%] was less than 1 cell/μL, and 18 patients had counts of 0 cells/μL. At the 6-month follow-up, the rituximab and obinutuzumab groups had no significant differences in immunological remission (80% vs 64%; OR: 2.29 [0.62– 8.47]; P=0.211) or clinical remission (76% vs 59%; OR: 2.19 [0.63– 7.66]; P=0.215]. No patients experienced serious adverse events.Conclusion: This retrospective analysis suggests that obinutuzumab may have potential as an initial therapeutic option for patients with PMN, although larger controlled studies are needed for confirmation.Keywords: obinutuzumab, PLA2R, membranous nephropathy, proteinuria
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spelling doaj-art-bfde803474a94013a11cc8d1e116ba0f2025-08-20T03:11:45ZengDove Medical PressDrug Design, Development and Therapy1177-88812025-07-01Volume 19Issue 159615972104720Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center TrialLi XQ0Liu Y1Cai ZY2Lv TG3Hao J4Department of Medicine, Division of NephrologyDepartment of Medicine, Division of NephrologyDepartment of Medicine, Division of NephrologyDepartment of Medicine, Division of RadiologyDepartment of Medicine, Division of NephrologyXue-Qi Li,1 Yang Liu,1 Ze-Yu Cai,1 Tie-Gang Lv,2 Jian Hao1 1Department of Medicine, Division of Nephrology, The Affiliated Hospital of Inner Mongolia Medical University, Hohhot, Inner Mongolia Autonomous Region, 010050, China; 2Department of Medicine, Division of Radiology, The Affiliated Hospital of Inner Mongolia Medical University, Hohhot, Inner Mongolia Autonomous Region, 010050, People’s Republic of ChinaCorrespondence: Jian Hao, Department of Medicine, Division of Nephrology, The Affiliated Hospital of Inner Mongolia Medical University, No. 1 North Passage Road, Huimin District, Hohhot, Inner Mongolia Autonomous Region, 010050, People’s Republic of China, Tel +8613704751021, Email jian_hao8865@126.comBackground: Membranous nephropathy (MN) can cause nephrotic syndrome. B cells contribute to MN, but available treatments are often inadequate. We addressed this treatment gap by analyzing the effect of obinutuzumab in patients with primary MN (PMN).Methods: Forty-seven PMN patients were followed for six months, with 25 receiving obinutuzumab and 22 (control) receiving rituximab. Treatment response was assessed by 24-h urine total protein (24-h UTP), serum albumin (ALB), and other indicators. Immunologic remission was assessed by measurement of anti-phospholipase A2 receptor autoantibodies (PLA2R autoAbs).Results: Relative to baseline, the obinutuzumab group had significant decreases of PLA2R autoAbs (83.40 [55.90– 344.36] vs 0.41 [0.17– 1.20] RU/mL), 24-h UTP (8.90 [7.15– 13.80) vs 1.82 [1.12– 3.43] g/day), and B cells (312.61 [202.00– 406.12) vs 0 [0– 0] cells/μL), and a significant increase of serum ALB (25.90 [20.85– 28.70] vs 42 [39.7– 45.3] g/L) after six months. Nineteen of the evaluable patients (76% [55– 91%]) achieved immunological remission at three months, 20 (80% [60– 93%] achieved immunological remission at six months, and 16 (64% [42– 83%] achieved partial response (PR) at three-months. After six-months, no patients achieved complete remission, but 19 (76% [55– 91%]) achieved PR. Before the second dose of obinutuzumab, the CD19+ B cell count in 20 patients (80%) [60%– 93%] was less than 1 cell/μL, and 18 patients had counts of 0 cells/μL. At the 6-month follow-up, the rituximab and obinutuzumab groups had no significant differences in immunological remission (80% vs 64%; OR: 2.29 [0.62– 8.47]; P=0.211) or clinical remission (76% vs 59%; OR: 2.19 [0.63– 7.66]; P=0.215]. No patients experienced serious adverse events.Conclusion: This retrospective analysis suggests that obinutuzumab may have potential as an initial therapeutic option for patients with PMN, although larger controlled studies are needed for confirmation.Keywords: obinutuzumab, PLA2R, membranous nephropathy, proteinuriahttps://www.dovepress.com/obinutuzumab-is-effective-as-an-initial-treatment-for-pla2r-associated-peer-reviewed-fulltext-article-DDDTObinutuzumabPLA2Rmembranous nephropathyproteinuria
spellingShingle Li XQ
Liu Y
Cai ZY
Lv TG
Hao J
Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center Trial
Drug Design, Development and Therapy
Obinutuzumab
PLA2R
membranous nephropathy
proteinuria
title Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center Trial
title_full Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center Trial
title_fullStr Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center Trial
title_full_unstemmed Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center Trial
title_short Obinutuzumab is Effective as an Initial Treatment for PLA2R-Associated Primary Membranous Nephropathy: A Retrospective, Single-Center Trial
title_sort obinutuzumab is effective as an initial treatment for pla2r associated primary membranous nephropathy a retrospective single center trial
topic Obinutuzumab
PLA2R
membranous nephropathy
proteinuria
url https://www.dovepress.com/obinutuzumab-is-effective-as-an-initial-treatment-for-pla2r-associated-peer-reviewed-fulltext-article-DDDT
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