Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cells

Aging is a physiological process that leads to degeneration and functional decline of the brain. This is accompanied by intracellular peroxidation and neuronal apoptosis. Natural antioxidants possess a remarkable effect on attenuating the oxidative stress cascade and apoptosis of neurons; however, t...

Full description

Saved in:
Bibliographic Details
Main Authors: Xiaoyu Xia, Han Li, Xianbing Xu, Zhenyu Wang, Junjie Yi, Guanghua Zhao, Ming Du
Format: Article
Language:English
Published: Tsinghua University Press 2025-03-01
Series:Food Science and Human Wellness
Subjects:
Online Access:https://www.sciopen.com/article/10.26599/FSHW.2024.9250057
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850096448205488128
author Xiaoyu Xia
Han Li
Xianbing Xu
Zhenyu Wang
Junjie Yi
Guanghua Zhao
Ming Du
author_facet Xiaoyu Xia
Han Li
Xianbing Xu
Zhenyu Wang
Junjie Yi
Guanghua Zhao
Ming Du
author_sort Xiaoyu Xia
collection DOAJ
description Aging is a physiological process that leads to degeneration and functional decline of the brain. This is accompanied by intracellular peroxidation and neuronal apoptosis. Natural antioxidants possess a remarkable effect on attenuating the oxidative stress cascade and apoptosis of neurons; however, the challenge of using natural antioxidants for neuroprotection is fabricating a delivery system to overcome the blood-brain barrier (BBB) transport. Herein, we successfully created a stable delivery platform built on rigid ferritin nanocage loading natural lycopene molecules, crossing the BBB in quantity and being taken up in neurons. This nanoparticle worked on D-galactose-induced senescence via alleviating neuronal hyperoxidation injury and weakening neuronal apoptosis in PC12 and BV2 cells. More importantly, this natural delivery system possesses inherent biocompatibility and potential application in improving the bioavailability of bioactive edible compounds with low water solubility. This study demonstrated the effectiveness of natural antioxidant nanomedicines in maintaining the defenses of intracerebral peroxidation and improve degenerating neurons, providing the potential to combat further imbalances of neuronal microenvironment in aging neuropathy.
format Article
id doaj-art-b50de17d93ac4d90bafd6030909d72ec
institution DOAJ
issn 2097-0765
2213-4530
language English
publishDate 2025-03-01
publisher Tsinghua University Press
record_format Article
series Food Science and Human Wellness
spelling doaj-art-b50de17d93ac4d90bafd6030909d72ec2025-08-20T02:41:14ZengTsinghua University PressFood Science and Human Wellness2097-07652213-45302025-03-01143925005710.26599/FSHW.2024.9250057Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cellsXiaoyu Xia0Han Li1Xianbing Xu2Zhenyu Wang3Junjie Yi4Guanghua Zhao5Ming Du6School of Food Science and Technology, Dalian Polytechnic University, Dalian 116034, ChinaSchool of Food Science and Technology, Dalian Polytechnic University, Dalian 116034, ChinaSchool of Food Science and Technology, Dalian Polytechnic University, Dalian 116034, ChinaSchool of Food Science and Technology, Dalian Polytechnic University, Dalian 116034, ChinaFaculty of Food Science and Engineering, Kunming University of Science and Technology, Kunming 650500, ChinaCollege of Food Science and Nutritional Engineering, China Agricultural University, Beijing 100083, ChinaSchool of Food Science and Technology, Dalian Polytechnic University, Dalian 116034, ChinaAging is a physiological process that leads to degeneration and functional decline of the brain. This is accompanied by intracellular peroxidation and neuronal apoptosis. Natural antioxidants possess a remarkable effect on attenuating the oxidative stress cascade and apoptosis of neurons; however, the challenge of using natural antioxidants for neuroprotection is fabricating a delivery system to overcome the blood-brain barrier (BBB) transport. Herein, we successfully created a stable delivery platform built on rigid ferritin nanocage loading natural lycopene molecules, crossing the BBB in quantity and being taken up in neurons. This nanoparticle worked on D-galactose-induced senescence via alleviating neuronal hyperoxidation injury and weakening neuronal apoptosis in PC12 and BV2 cells. More importantly, this natural delivery system possesses inherent biocompatibility and potential application in improving the bioavailability of bioactive edible compounds with low water solubility. This study demonstrated the effectiveness of natural antioxidant nanomedicines in maintaining the defenses of intracerebral peroxidation and improve degenerating neurons, providing the potential to combat further imbalances of neuronal microenvironment in aging neuropathy.https://www.sciopen.com/article/10.26599/FSHW.2024.9250057ferritinlycopenenanocarrierneuroprotectionaging
spellingShingle Xiaoyu Xia
Han Li
Xianbing Xu
Zhenyu Wang
Junjie Yi
Guanghua Zhao
Ming Du
Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cells
Food Science and Human Wellness
ferritin
lycopene
nanocarrier
neuroprotection
aging
title Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cells
title_full Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cells
title_fullStr Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cells
title_full_unstemmed Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cells
title_short Ferritin nanocage loading lycopene for improving blood-brain barrier transcytosis and attenuating D-galactose-induced apoptosis in PC12 cells
title_sort ferritin nanocage loading lycopene for improving blood brain barrier transcytosis and attenuating d galactose induced apoptosis in pc12 cells
topic ferritin
lycopene
nanocarrier
neuroprotection
aging
url https://www.sciopen.com/article/10.26599/FSHW.2024.9250057
work_keys_str_mv AT xiaoyuxia ferritinnanocageloadinglycopeneforimprovingbloodbrainbarriertranscytosisandattenuatingdgalactoseinducedapoptosisinpc12cells
AT hanli ferritinnanocageloadinglycopeneforimprovingbloodbrainbarriertranscytosisandattenuatingdgalactoseinducedapoptosisinpc12cells
AT xianbingxu ferritinnanocageloadinglycopeneforimprovingbloodbrainbarriertranscytosisandattenuatingdgalactoseinducedapoptosisinpc12cells
AT zhenyuwang ferritinnanocageloadinglycopeneforimprovingbloodbrainbarriertranscytosisandattenuatingdgalactoseinducedapoptosisinpc12cells
AT junjieyi ferritinnanocageloadinglycopeneforimprovingbloodbrainbarriertranscytosisandattenuatingdgalactoseinducedapoptosisinpc12cells
AT guanghuazhao ferritinnanocageloadinglycopeneforimprovingbloodbrainbarriertranscytosisandattenuatingdgalactoseinducedapoptosisinpc12cells
AT mingdu ferritinnanocageloadinglycopeneforimprovingbloodbrainbarriertranscytosisandattenuatingdgalactoseinducedapoptosisinpc12cells