A zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation

Abstract Borylation chemistry plays a crucial role in the development of new synthetic methodologies. However, the reactivity of zinc-boryl species has not been fully explored, particularly in relation to diverse reaction pathways. Here we show that a zinc-boryl species is successfully synthesized f...

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Main Authors: Gan Xu, Hok Tsun Chan, Shuchang Li, Tsz Ying Wong, Lei Zhang, Qichun Zhang, Zhenyang Lin, Zhenpin Lu
Format: Article
Language:English
Published: Nature Portfolio 2025-07-01
Series:Nature Communications
Online Access:https://doi.org/10.1038/s41467-025-61062-z
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author Gan Xu
Hok Tsun Chan
Shuchang Li
Tsz Ying Wong
Lei Zhang
Qichun Zhang
Zhenyang Lin
Zhenpin Lu
author_facet Gan Xu
Hok Tsun Chan
Shuchang Li
Tsz Ying Wong
Lei Zhang
Qichun Zhang
Zhenyang Lin
Zhenpin Lu
author_sort Gan Xu
collection DOAJ
description Abstract Borylation chemistry plays a crucial role in the development of new synthetic methodologies. However, the reactivity of zinc-boryl species has not been fully explored, particularly in relation to diverse reaction pathways. Here we show that a zinc-boryl species is successfully synthesized from bis(catecholato)diboron, exhibiting amphiphilic reactivity. This compound acts as a nucleophilic boron anion with methyl iodide and as an electrophile with N,N’-dicyclohexylcarbodiimide, facilitating zinc-boron bond dissociation and generating zinc-carbon and zinc-nitrogen bonds while cleaving carbon-nitrogen double bonds. The enhanced reactivity is likely due to the stronger covalency of the zinc-boron bond. Additionally, the zinc-boryl compound promotes the catalytic diborylation of azobenzene, underscoring its versatility as a reactive intermediate. Density functional theory studies illuminate the electronic structure and reactivity of the zinc-boron bond, providing insights into potential applications in synthetic chemistry.
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id doaj-art-a351389e2a1b4aaba5b1fc98da660b18
institution Kabale University
issn 2041-1723
language English
publishDate 2025-07-01
publisher Nature Portfolio
record_format Article
series Nature Communications
spelling doaj-art-a351389e2a1b4aaba5b1fc98da660b182025-08-20T03:43:27ZengNature PortfolioNature Communications2041-17232025-07-011611810.1038/s41467-025-61062-zA zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylationGan Xu0Hok Tsun Chan1Shuchang Li2Tsz Ying Wong3Lei Zhang4Qichun Zhang5Zhenyang Lin6Zhenpin Lu7Department of Chemistry, State Key Laboratory of Marine Pollution, City University of Hong KongDepartment of Chemistry, The Hong Kong University of Science and TechnologyDepartment of Chemistry, State Key Laboratory of Marine Pollution, City University of Hong KongDepartment of Chemistry, State Key Laboratory of Marine Pollution, City University of Hong KongDepartment of Materials Science and Engineering, City University of Hong KongDepartment of Materials Science and Engineering, City University of Hong KongDepartment of Chemistry, The Hong Kong University of Science and TechnologyDepartment of Chemistry, State Key Laboratory of Marine Pollution, City University of Hong KongAbstract Borylation chemistry plays a crucial role in the development of new synthetic methodologies. However, the reactivity of zinc-boryl species has not been fully explored, particularly in relation to diverse reaction pathways. Here we show that a zinc-boryl species is successfully synthesized from bis(catecholato)diboron, exhibiting amphiphilic reactivity. This compound acts as a nucleophilic boron anion with methyl iodide and as an electrophile with N,N’-dicyclohexylcarbodiimide, facilitating zinc-boron bond dissociation and generating zinc-carbon and zinc-nitrogen bonds while cleaving carbon-nitrogen double bonds. The enhanced reactivity is likely due to the stronger covalency of the zinc-boron bond. Additionally, the zinc-boryl compound promotes the catalytic diborylation of azobenzene, underscoring its versatility as a reactive intermediate. Density functional theory studies illuminate the electronic structure and reactivity of the zinc-boron bond, providing insights into potential applications in synthetic chemistry.https://doi.org/10.1038/s41467-025-61062-z
spellingShingle Gan Xu
Hok Tsun Chan
Shuchang Li
Tsz Ying Wong
Lei Zhang
Qichun Zhang
Zhenyang Lin
Zhenpin Lu
A zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation
Nature Communications
title A zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation
title_full A zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation
title_fullStr A zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation
title_full_unstemmed A zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation
title_short A zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation
title_sort zinc boryl compound unlocks diverse reactivity pathways beyond nucleophilic borylation
url https://doi.org/10.1038/s41467-025-61062-z
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