5-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cells

5-Aminolevulinic acid hydrochloride (ALA)-mediated sonodynamic therapy (SDT) had anti-tumour effect on pancreatic cancer cells. Hence, ALA loaded lipid/poly(lactic-co-glycolic acid) (PLGA) microbubbles (MBs)-mediated SDT for pancreatic cancer has great potential. The average size of ALA-lipid MBs an...

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Main Authors: Wei Yang, Haitao Xu, Qinghao Liu, Chunxun Liu, Jiahe Hu, Ping Liu, Tianyi Fang, Yuxian Bai, Jiuxin Zhu, Rui Xie
Format: Article
Language:English
Published: Taylor & Francis Group 2020-01-01
Series:Artificial Cells, Nanomedicine, and Biotechnology
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Online Access:https://www.tandfonline.com/doi/10.1080/21691401.2020.1813743
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author Wei Yang
Haitao Xu
Qinghao Liu
Chunxun Liu
Jiahe Hu
Ping Liu
Tianyi Fang
Yuxian Bai
Jiuxin Zhu
Rui Xie
author_facet Wei Yang
Haitao Xu
Qinghao Liu
Chunxun Liu
Jiahe Hu
Ping Liu
Tianyi Fang
Yuxian Bai
Jiuxin Zhu
Rui Xie
author_sort Wei Yang
collection DOAJ
description 5-Aminolevulinic acid hydrochloride (ALA)-mediated sonodynamic therapy (SDT) had anti-tumour effect on pancreatic cancer cells. Hence, ALA loaded lipid/poly(lactic-co-glycolic acid) (PLGA) microbubbles (MBs)-mediated SDT for pancreatic cancer has great potential. The average size of ALA-lipid MBs and ALA-PLGA MBs was about 3.0 µm. The two kinds of MBs had good biocompatibility to normal HPDE6-C7 cells and were not toxic to pancreatic cancer cells. Compared with ALA-induced SDT, a statistically significant decrease in cell viability was observed in ALA lipid/PLGA MBs combined with ultrasound groups in AsPC-1 and BxPC-3 cells (p < .05). Obvious effect on the apoptotic rate, apoptosis and pyroptosis morphology, enhanced reactive oxygen species was found in ALA-lipid/PLGA MBs mediated SDT in vitro. Through in vivo study, we found ALA-lipid/PLGA MBs-mediated SDT was a promise treatment for pancreatic cancer.
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institution Kabale University
issn 2169-1401
2169-141X
language English
publishDate 2020-01-01
publisher Taylor & Francis Group
record_format Article
series Artificial Cells, Nanomedicine, and Biotechnology
spelling doaj-art-6e7d03bc97da4562a9d1e7c3c2ebc9c82025-08-20T03:41:25ZengTaylor & Francis GroupArtificial Cells, Nanomedicine, and Biotechnology2169-14012169-141X2020-01-014811178118810.1080/21691401.2020.18137435-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cellsWei Yang0Haitao Xu1Qinghao Liu2Chunxun Liu3Jiahe Hu4Ping Liu5Tianyi Fang6Yuxian Bai7Jiuxin Zhu8Rui Xie9Harbin Medical University Cancer Hospital, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, ChinaDepartment of Pharmacology (State-Province Key Laboratories of Biomedicine-Pharmaceutics of China, Key Laboratories of Cardiovascular Medicine Research, Ministry of Education), College of Pharmacy, Harbin Medical University, Harbin, ChinaHarbin Medical University Cancer Hospital, Harbin, China5-Aminolevulinic acid hydrochloride (ALA)-mediated sonodynamic therapy (SDT) had anti-tumour effect on pancreatic cancer cells. Hence, ALA loaded lipid/poly(lactic-co-glycolic acid) (PLGA) microbubbles (MBs)-mediated SDT for pancreatic cancer has great potential. The average size of ALA-lipid MBs and ALA-PLGA MBs was about 3.0 µm. The two kinds of MBs had good biocompatibility to normal HPDE6-C7 cells and were not toxic to pancreatic cancer cells. Compared with ALA-induced SDT, a statistically significant decrease in cell viability was observed in ALA lipid/PLGA MBs combined with ultrasound groups in AsPC-1 and BxPC-3 cells (p < .05). Obvious effect on the apoptotic rate, apoptosis and pyroptosis morphology, enhanced reactive oxygen species was found in ALA-lipid/PLGA MBs mediated SDT in vitro. Through in vivo study, we found ALA-lipid/PLGA MBs-mediated SDT was a promise treatment for pancreatic cancer.https://www.tandfonline.com/doi/10.1080/21691401.2020.1813743Pancreatic cancersonodynamic therapy5-aminolevulinic acidmicrobubblesapoptosispyroptosis
spellingShingle Wei Yang
Haitao Xu
Qinghao Liu
Chunxun Liu
Jiahe Hu
Ping Liu
Tianyi Fang
Yuxian Bai
Jiuxin Zhu
Rui Xie
5-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cells
Artificial Cells, Nanomedicine, and Biotechnology
Pancreatic cancer
sonodynamic therapy
5-aminolevulinic acid
microbubbles
apoptosis
pyroptosis
title 5-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cells
title_full 5-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cells
title_fullStr 5-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cells
title_full_unstemmed 5-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cells
title_short 5-Aminolevulinic acid hydrochloride loaded microbubbles-mediated sonodynamic therapy in pancreatic cancer cells
title_sort 5 aminolevulinic acid hydrochloride loaded microbubbles mediated sonodynamic therapy in pancreatic cancer cells
topic Pancreatic cancer
sonodynamic therapy
5-aminolevulinic acid
microbubbles
apoptosis
pyroptosis
url https://www.tandfonline.com/doi/10.1080/21691401.2020.1813743
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