Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro Study

Background: Vitamin E, a fat-soluble vitamin, protects cell membranes by scavenging free radicals and reducing lipid peroxidation. It plays a crucial role in immune cell function, gene expression, and modulation of inflammatory mediators. Nanoparticles in drug delivery, particularly chitosan-based n...

Full description

Saved in:
Bibliographic Details
Main Authors: Turaga Amani, Mouttoukichenin Surenthar
Format: Article
Language:English
Published: Wolters Kluwer Medknow Publications 2025-01-01
Series:Journal of Indian Academy of Oral Medicine and Radiology
Subjects:
Online Access:https://journals.lww.com/10.4103/jiaomr.jiaomr_265_24
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850203196818980864
author Turaga Amani
Mouttoukichenin Surenthar
author_facet Turaga Amani
Mouttoukichenin Surenthar
author_sort Turaga Amani
collection DOAJ
description Background: Vitamin E, a fat-soluble vitamin, protects cell membranes by scavenging free radicals and reducing lipid peroxidation. It plays a crucial role in immune cell function, gene expression, and modulation of inflammatory mediators. Nanoparticles in drug delivery, particularly chitosan-based nanogels, enhance solubility and prolong biological activity. Objective: This study aims to evaluate the antioxidant and anti-inflammatory activity of a vitamin E-infused nanogel formulation in an in-vitro setting and compare its efficacy with standard antioxidant and anti-inflammatory agents. Methods: A gel was created by lyophilizing 5 g of powdered vitamin E, 0.5 g of chitosan, 0.2 mL of tween 80, and 10 mL of monosodium phosphate in 90 mL of distilled water, which was then heated to 55°C for 30 minutes while stirring. The formulation’s antioxidant and anti-inflammatory activities were assessed using standard assays, such as DPPH (2,2-diphenyl-1-picrylhydrazyl) radical scavenging and albumin denaturation assays. The nanogel’s effectiveness was assessed by comparing its percentage inhibition values at different concentrations with those of standard antioxidants (ascorbic acid) and anti-inflammatory agents (diclofenac sodium). Results: The vitamin E-infused nanogel demonstrated antioxidant and anti-inflammatory properties comparable to standard drugs, with the highest activity observed at 100 µg/mL in both assays. Conclusion: The study demonstrates that the vitamin E-infused nanogel exhibits promising in-vitro antioxidant and anti-inflammatory activities, with inhibition percentages comparable to standard drugs. Further validation through statistical analysis and in-vivo studies is required to confirm its therapeutic potential in managing oral potentially malignant disorders.
format Article
id doaj-art-4dcb45ba9ef4491ebe9aa8c204345a1d
institution OA Journals
issn 0972-1363
0975-1572
language English
publishDate 2025-01-01
publisher Wolters Kluwer Medknow Publications
record_format Article
series Journal of Indian Academy of Oral Medicine and Radiology
spelling doaj-art-4dcb45ba9ef4491ebe9aa8c204345a1d2025-08-20T02:11:34ZengWolters Kluwer Medknow PublicationsJournal of Indian Academy of Oral Medicine and Radiology0972-13630975-15722025-01-01371788210.4103/jiaomr.jiaomr_265_24Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro StudyTuraga AmaniMouttoukichenin SurentharBackground: Vitamin E, a fat-soluble vitamin, protects cell membranes by scavenging free radicals and reducing lipid peroxidation. It plays a crucial role in immune cell function, gene expression, and modulation of inflammatory mediators. Nanoparticles in drug delivery, particularly chitosan-based nanogels, enhance solubility and prolong biological activity. Objective: This study aims to evaluate the antioxidant and anti-inflammatory activity of a vitamin E-infused nanogel formulation in an in-vitro setting and compare its efficacy with standard antioxidant and anti-inflammatory agents. Methods: A gel was created by lyophilizing 5 g of powdered vitamin E, 0.5 g of chitosan, 0.2 mL of tween 80, and 10 mL of monosodium phosphate in 90 mL of distilled water, which was then heated to 55°C for 30 minutes while stirring. The formulation’s antioxidant and anti-inflammatory activities were assessed using standard assays, such as DPPH (2,2-diphenyl-1-picrylhydrazyl) radical scavenging and albumin denaturation assays. The nanogel’s effectiveness was assessed by comparing its percentage inhibition values at different concentrations with those of standard antioxidants (ascorbic acid) and anti-inflammatory agents (diclofenac sodium). Results: The vitamin E-infused nanogel demonstrated antioxidant and anti-inflammatory properties comparable to standard drugs, with the highest activity observed at 100 µg/mL in both assays. Conclusion: The study demonstrates that the vitamin E-infused nanogel exhibits promising in-vitro antioxidant and anti-inflammatory activities, with inhibition percentages comparable to standard drugs. Further validation through statistical analysis and in-vivo studies is required to confirm its therapeutic potential in managing oral potentially malignant disorders.https://journals.lww.com/10.4103/jiaomr.jiaomr_265_24anti-inflammatory agentsantioxidantschitosannanoparticle drug delivery systemvitamin e
spellingShingle Turaga Amani
Mouttoukichenin Surenthar
Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro Study
Journal of Indian Academy of Oral Medicine and Radiology
anti-inflammatory agents
antioxidants
chitosan
nanoparticle drug delivery system
vitamin e
title Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro Study
title_full Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro Study
title_fullStr Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro Study
title_full_unstemmed Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro Study
title_short Anti-Inflammatory and Antioxidant Activity of Vitamin E-infused Nanogel Formulation: An In-Vitro Study
title_sort anti inflammatory and antioxidant activity of vitamin e infused nanogel formulation an in vitro study
topic anti-inflammatory agents
antioxidants
chitosan
nanoparticle drug delivery system
vitamin e
url https://journals.lww.com/10.4103/jiaomr.jiaomr_265_24
work_keys_str_mv AT turagaamani antiinflammatoryandantioxidantactivityofvitamineinfusednanogelformulationaninvitrostudy
AT mouttoukicheninsurenthar antiinflammatoryandantioxidantactivityofvitamineinfusednanogelformulationaninvitrostudy