The human ABCG2 transporter engages three gates to control multidrug extrusion

Summary: The human ABCG2 transporter plays roles in physiological detoxification across barriers and in anticancer multidrug resistance. The translocation pathway for drug extrusion and its gating mechanism remains elusive. Here, we demonstrate that the ABCG2 multidrug transporter holds two cavities...

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Bibliographic Details
Main Authors: Narakorn Khunweeraphong, Karl Kuchler
Format: Article
Language:English
Published: Elsevier 2025-03-01
Series:iScience
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S2589004225003852
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