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Crystal structures of Mycobacterium tuberculosis and Mycobacterium thermoresistibile glycyl-tRNA synthetases in various liganded states. by Michael K Fenwick, Amy E DeRocher, Justin K Craig, Elizabeth K Harmon, Steve Seibold, Lijun Liu, Kevin P Battaile, Lynn K Barrett, Wesley C Van Voorhis, Isabelle Q Phan, Bart L Staker, Sandhya Subramanian, Scott Lovell, Peter J Myler
Published 2025-01-01Get full text
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High-throughput screening of the ReFRAME, Pandemic Box, and COVID Box drug repurposing libraries against SARS-CoV-2 nsp15 endoribonuclease to identify small-molecule inhibitors of... by Ryan Choi, Mowei Zhou, Roger Shek, Jesse W Wilson, Logan Tillery, Justin K Craig, Indraneel A Salukhe, Sarah E Hickson, Neeraj Kumar, Rhema M James, Garry W Buchko, Ruilian Wu, Sydney Huff, Tu-Trinh Nguyen, Brett L Hurst, Sara Cherry, Lynn K Barrett, Jennifer L Hyde, Wesley C Van Voorhis
Published 2021-01-01Get full text
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Anti-Cryptosporidium efficacy of BKI-1708, an inhibitor of Cryptosporidium calcium-dependent protein kinase 1. by Ryan Choi, Matthew A Hulverson, Deborah A Schaefer, Dana P Betzer, Michael W Riggs, Wenlin Huang, Vicky Sun, Grant R Whitman, Molly C McCloskey, Kennan Marsh, Wayne R Buck, David S Wagner, Junhai Yang, Andrew P Bowman, Rita Ciurlionis, Jubilee Ajiboye, Andrew Hemphill, Dilep K Sigalapalli, Samuel L M Arnold, Lynn K Barrett, Kayode K Ojo, Erkang Fan, Wesley C Van Voorhis
Published 2025-07-01Get full text
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Anti-Cryptosporidium efficacy of BKI-1708, an inhibitor of Cryptosporidium calcium-dependent protein kinase 1 by Ryan Choi, Matthew A. Hulverson, Deborah A. Schaefer, Dana P. Betzer, Michael W. Riggs, Wenlin Huang, Vicky Sun, Grant R. Whitman, Molly C. McCloskey, Kennan Marsh, Wayne R. Buck, David S. Wagner, Junhai Yang, Andrew P. Bowman, Rita Ciurlionis, Jubilee Ajiboye, Andrew Hemphill, Dilep K. Sigalapalli, Samuel L.M. Arnold, Lynn K. Barrett, Kayode K. Ojo, Erkang Fan, Wesley C. Van Voorhis
Published 2025-07-01Get full text
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5
Naegleria fowleri: Protein structures to facilitate drug discovery for the deadly, pathogenic free-living amoeba. by Logan Tillery, Kayleigh Barrett, Jenna Goldstein, Jared W Lassner, Bram Osterhout, Nathan L Tran, Lily Xu, Ryan M Young, Justin Craig, Ian Chun, David M Dranow, Jan Abendroth, Silvia L Delker, Douglas R Davies, Stephen J Mayclin, Brandy Calhoun, Madison J Bolejack, Bart Staker, Sandhya Subramanian, Isabelle Phan, Donald D Lorimer, Peter J Myler, Thomas E Edwards, Dennis E Kyle, Christopher A Rice, James C Morris, James W Leahy, Roman Manetsch, Lynn K Barrett, Craig L Smith, Wesley C Van Voorhis
Published 2021-01-01Get full text
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Exquisite selectivity of griselimycin extends to beta subunit of DNA polymerases from Gram-negative bacterial pathogens by Michael K. Fenwick, Phillip G. Pierce, Jan Abendroth, Kayleigh F. Barrett, Lynn K. Barrett, Kalinga Bowatte, Ryan Choi, Ian Chun, Deborah G. Conrady, Justin K. Craig, David M. Dranow, Bradley Hammerson, Tate Higgins, Donald D. Lorimer, Peer Lukat, Stephen J. Mayclin, Stephen Nakazawa Hewitt, Ying Po Peng, Ashwini Shanbhogue, Hayden Smutney, Matthew Z. Z. Stigliano, Logan M. Tillery, Hannah S. Udell, Ellen G. Wallace, Amy E. DeRocher, Isabelle Q. Phan, Bart L. Staker, Sandhya Subramanian, Wesley C. Van Voorhis, Wulf Blankenfeldt, Rolf Müller, Thomas E. Edwards, Peter J. Myler
Published 2024-12-01Get full text
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