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A novel 4-aminoquinoline chemotype with multistage antimalarial activity and lack of cross-resistance with PfCRT and PfMDR1 mutants. by Letícia Tiburcio Ferreira, Gustavo Capatti Cassiano, Luis Carlos Salazar Alvarez, John Okombo, Juliana Calit, Diana Fontinha, Eva Gil-Iturbe, Rachael Coyle, Carolina Horta Andrade, Per Sunnerhagen, Daniel Youssef Bargieri, Miguel Prudêncio, Matthias Quick, Pedro V Cravo, Marcus C S Lee, David A Fidock, Fabio Trindade Maranhão Costa
Published 2024-10-01Get full text
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Pyrimidine Azepine Targets the Plasmodium bc1 Complex and Displays Multistage Antimalarial Activity by Juliana Calit, Surendra K. Prajapati, Ernest D. Benavente, Jessica E. Araújo, Bingbing Deng, Kazutoyo Miura, Yasmin Annunciato, Igor M. R. Moura, Miho Usui, Jansen F. Medeiros, Carolina H. Andrade, Sabrina Silva-Mendonça, Anton Simeonov, Richard T. Eastman, Carole A. Long, Maisa da Silva Araujo, Kim C. Williamson, Anna Caroline C. Aguiar, Daniel Y. Bargieri
Published 2024-10-01Get full text
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