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Development of novel pyrimidine-thio-triazoles targeting EGFR in breast Cancer cells via one-pot copper-catalyzed 1,3-dipolar cycloaddition by Bhanuprakash C. Narasimhachar, Akshay Ravish, Narasimha M. Beeraka, Baburajeev Chumadathil Pookunoth, Shreeja Basappa, Divakar Vishwanath, Kanchugarakoppal S. Rangappa, Omantheswara Nagaraja, Mahendra Madegowda, Paduvalahippe Gowdegowda Chandrashekara, Basappa Basappa
Published 2025-03-01Get full text
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Discovery of 2‑Pyrazolines That Inhibit the Phosphorylation of STAT3 as Nanomolar Cytotoxic Agents by Tejaswini P. Siddappa, Akshay Ravish, Zhang Xi, Arunkumar Mohan, Swamy S. Girimanchanaika, Niranjan Pattehali Krishnamurthy, Shreeja Basappa, Santosh L. Gaonkar, Peter E. Lobie, Vijay Pandey, Basappa Basappa
Published 2025-01-01Get full text
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Dual action of pyrimidine derivatives: Targeting tamoxifen resistance in breast cancer by Jie Yuan, Geng Wang, Narasimha M. Beeraka, Hua Zhang, Qun Wang, Danfeng Zhang, Minghua Wang, Akshay Ravish, Arunachalam Chinnathambi, Sulaiman Ali Alharbi, Kanchugarakoppal S. Rangappa, Vladimir N. Nikolenko, Basappa Basappa, Li Yang
Published 2025-08-01Get full text
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A novel drug prejudice scaffold-imidazopyridine-conjugate can promote cell death in a colorectal cancer model by binding to β-catenin and suppressing the Wnt signaling pathway by Min Hee Yang, Basappa Basappa, Suresha N. Deveshegowda, Akshay Ravish, Arunkumar Mohan, Omantheswara Nagaraja, Mahendra Madegowda, Kanchugarakoppal S. Rangappa, Amudha Deivasigamani, Vijay Pandey, Peter E. Lobie, Kam Man Hui, Gautam Sethi, Kwang Seok Ahn
Published 2025-06-01Get full text
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